Synthesis of irreversibly binding bicalutamide analogs for imaging studies

Vipin A. Nair; Suni M. Mustafa; Michael L. Mohler; Jun Yang; Leonid I. Kirkovsky; James T. Dalton; Duane D. Miller

doi:10.1016/j.tetlet.2005.04.143

Synthesis of irreversibly binding bicalutamide analogs for imaging studies

Vipin A. Nair, Suni M. Mustafa, Michael L. Mohler, Jun Yang, Leonid I. Kirkovsky, James T. Dalton, Duane D. Miller^*

^*Corresponding author for this work

Research output: Contribution to journal › Article › peer-review

12 Citations (Scopus)

Abstract

A new synthetic methodology for preparing radioactive androgen receptor binding compounds in order to determine receptor-ligands interactions has been developed.

Original language	English
Pages (from-to)	4821-4823
Number of pages	3
Journal	Tetrahedron Letters
Volume	46
Issue number	28
DOIs	https://doi.org/10.1016/j.tetlet.2005.04.143
Publication status	Published - 11 Jul 2005
Externally published	Yes

Keywords

Androgen
Bicalutamide
Iodine
Radioactive
Receptor

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10.1016/j.tetlet.2005.04.143

Cite this

@article{30e9cc2423c24b8daf4dd2acac2f9b06,

title = "Synthesis of irreversibly binding bicalutamide analogs for imaging studies",

abstract = "A new synthetic methodology for preparing radioactive androgen receptor binding compounds in order to determine receptor-ligands interactions has been developed.",

keywords = "Androgen, Bicalutamide, Iodine, Radioactive, Receptor",

author = "Nair, {Vipin A.} and Mustafa, {Suni M.} and Mohler, {Michael L.} and Jun Yang and Kirkovsky, {Leonid I.} and Dalton, {James T.} and Miller, {Duane D.}",

year = "2005",

month = jul,

day = "11",

doi = "10.1016/j.tetlet.2005.04.143",

language = "English",

volume = "46",

pages = "4821--4823",

journal = "Tetrahedron Letters",

issn = "0040-4039",

number = "28",

}

TY - JOUR

T1 - Synthesis of irreversibly binding bicalutamide analogs for imaging studies

AU - Nair, Vipin A.

AU - Mustafa, Suni M.

AU - Mohler, Michael L.

AU - Yang, Jun

AU - Kirkovsky, Leonid I.

AU - Dalton, James T.

AU - Miller, Duane D.

PY - 2005/7/11

Y1 - 2005/7/11

N2 - A new synthetic methodology for preparing radioactive androgen receptor binding compounds in order to determine receptor-ligands interactions has been developed.

AB - A new synthetic methodology for preparing radioactive androgen receptor binding compounds in order to determine receptor-ligands interactions has been developed.

KW - Androgen

KW - Bicalutamide

KW - Iodine

KW - Radioactive

KW - Receptor

UR - http://www.scopus.com/inward/record.url?scp=20444419774&partnerID=8YFLogxK

U2 - 10.1016/j.tetlet.2005.04.143

DO - 10.1016/j.tetlet.2005.04.143

M3 - Article

AN - SCOPUS:20444419774

SN - 0040-4039

VL - 46

SP - 4821

EP - 4823

JO - Tetrahedron Letters

JF - Tetrahedron Letters

IS - 28

ER -

Synthesis of irreversibly binding bicalutamide analogs for imaging studies

Abstract

Keywords

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